Structure Information
Structure

Compound Identification

SMILES

CCCCCN1C=NC2=CC=CC3=C2C1=C1CN2C(=CC4=C(COC(=O)[C@@]4(CC)OC(=O)CC[C@H](NC(=O)[C@@H](N)CCCCN)C(O)=O)C2=O)C1=N3

InChIKey

InChIKey=DKLPEWNIXJCAIA-QZDQGYFBSA-N

Formula

C37H45N7O8

Mass

715.808

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Taxonomic Classification

Taxonomy Tree

Kingdom

Organic compounds

Superclass

Alkaloids and derivatives

Class

Camptothecins

Subclass

Not available

Intermediate Tree Nodes

Not available

Direct Parent

Camptothecins

Alternative Parents

Molecular Framework

Aromatic heteropolycyclic compounds

Substituents

Camptothecin - Alpha-dipeptide - Alpha peptide - Glutamic acid or derivatives - N-acyl-alpha-amino acid - N-acyl-alpha amino acid or derivatives - N-acyl-l-alpha-amino acid - Alpha-amino acid amide - Diazanaphthalene - Alpha-amino acid or derivatives - Pyranopyridine - Pyridopyrimidine - Quinazoline - Quinoline - Tricarboxylic acid or derivatives - Fatty acid ester - Pyridinone - Fatty amide - Fatty acyl - Pyrimidine - N-acyl-amine - Benzenoid - Pyridine - Heteroaromatic compound - Lactam - Lactone - Carboxylic acid ester - Amino acid - Carboxamide group - Secondary carboxylic acid amide - Amino acid or derivatives - Carboxylic acid derivative - Carboxylic acid - Azacycle - Oxacycle - Organoheterocyclic compound - Organic oxygen compound - Organic nitrogen compound - Primary aliphatic amine - Hydrocarbon derivative - Organonitrogen compound - Carbonyl group - Organic oxide - Organooxygen compound - Amine - Primary amine - Aromatic heteropolycyclic compound

Description

This compound belongs to the class of organic compounds known as camptothecins. These are heterocyclic compounds comprising a planar pentacyclic ring structure, that includes a pyrrolo[3,4-beta]-quinoline moiety (rings A, B and C), conjugated pyridone moiety (ring D) and one chiral center at position 20 within the alpha-hydroxy lactone ring with (S) configuration (the E-ring).

External Descriptors

Not available

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